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GABA Receptor Activators

Cat.No. Product Name Information Product Use Citations Product Validations
S4423 Emamectin Benzoate Emamectin Benzoate (EMB, MK-244) activates gamma-amino butyric acid (GABA) transporter. This compound induces of reactive oxygen species (ROS)-mediated DNA damage and apoptosis.
Viruses, 2025, 17(2)220
S1969 Nefiracetam Nefiracetam (DZL 221) is a GABAergic, cholinergic, and monoaminergic neuronal system enhancer for Ro 5-4864-induced convulsions. Phase 2.
E3045 Chinese Arborvilea Seed Extract Chinese Arborvilea Seed Extract is extracted from the dried and mature seed kernels of Platycladus orientalis (L.)Franco, has obvious anti-anxiety effect, and its mechanism may be related to increasing GABA level and decreasing Glu level in hippocampus.
E2354 Valepotriate Valepotriate, an unstable iridoid isolated from Valeriana jatamansi Jones, has anti-epileptic by significantly increasing the expression of GABAA, glutamic acid Decarboxylase 65, and Bcl-2 and reduce the expression of caspase-3.
S4772 alpha-Asarone alpha-Asarone (trans-Asarone) is one of the main pharmacologically active compounds present in Acorus calamus Linn (Acoraceae), Acorus tatarinowii Schott (Acoraceae), and Acorus gramineus Solander. It has anticonvulsant, neuroprotective, anxiolytic and nootropic effects.
S5319 Imepitoin Imepitoin (ELB-138, AWD 131-138) is a centrally acting anti-epileptic which crosses the blood brain barrier and is used for the treatment of canine idiopathic epilepsy. This compound is an antiepileptic and antianxietic drug, it can stimulate different recombinant isoforms of the rat GABA(A) receptor through the benzodiazepine binding site.
S4494 Methionine Methionine (MRX-1024, D-Methionine) is an activator of GABAA receptor that modulates neuronal activity.