Home Neuronal Signaling -Transmembrane Transporters GABA Receptor GABAA receptor-Selective Agonists | Antagonists

GABAA receptor-Selective Agonists | Antagonists

  • GABAA receptor
  • GABAB receptor
Cat.No. Product Name Information Selective / Pan IC50 / Ki
S7071 (+)-Bicuculline (+)-Bicuculline is a competitive antagonist of GABAA receptors with IC50 of 2 μM, also blocks Ca(2+)-activated potassium channels. Selective GABAA receptor, IC50: 2 μM
S1332 Flumazenil Flumazenil is a competitive GABAA receptor antagonist, used in the treatment of benzodiazepine overdoses. Selective
S2399 Dihydromyricetin Dihydromyricetin (Ampelopsin, Ampeloptin) is a natural antioxidant flavonoid from Ampelopsis grossedentata. Selective
S2269 Baicalin Baicalin is a known prolyl endopeptidase inhibitor and affects the GABA receptors. Selective
S4197 Bemegride Bemegride is a central nervous system stimulant and antidote for barbiturate poisoning. Selective