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Bradykinin Receptor

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Cat.No. Product Name Information Product Use Citations Product Validations
S5695 Icatibant Acetate Icatibant Acetate (HOE-140 acetate) acts as an antagonist of the bradykinin B2 receptor and is used in the treatment of hereditary angioedema.
Kyushu University Institutional Repository, 2022,
E7418 Noscapine Noscapine ((S,R)-Noscapine) is an alkaloid derived from the opium poppy (Papaver somniferum) and is a centrally acting antitussive opiate derivative. It is a non-competitive antagonist of the bradykinin B2 receptor. This compound also exhibits neuroprotection by activating sigma-1 opioid receptors, which help suppress intracellular NO levels and calcium, thereby providing protection against ischaemic injury.
E0460 ELN441958 ELN-441958 is a potent, neutral, competitive and selective bradykinin B1 receptor antagonist with a Ki of 0.26 nM against native human bradykinin B1 receptor.